Multidimensional Pharmacochemistry: Design of Safer Drugs deals with techniques based on the theory of simultaneous statistical inference and the qualitative rules that can be applied in solving problems of high toxicity. This book points out that the multidimensional view of data analysis can be applied to solve problems in medicinal chemistry. Investigators use different approaches; a certain procedure can prove to be the most beneficial for a specific drug design. This text presents the theoretical assumptions that mathematicians make to derive the basis for their multivariate techniques. This book also describes, in nonmathematical terms, a set of methods that are valuable, as well as explain the different designs by using numerical examples. According to E.J. Ariens, drug action involves the pharmaceutical, pharmacokinetic-toxokinetic, and pharmacodynamics-toxodynamic phases. The multivariate structure-activity analysis (MASCA) Model of Pharmacochemistry is a highly unified multivariate approach to drug design. To develop a multidimensionally oriented pharmacology, the book notes that the investigator can use the "dynamic structure-activity analysis." This entails the experimentalist and chemist using quantitative approaches and intuitive elements from a small number of compounds toward larger groups, with successive changes being inputted in the desired biological activity. This book is strongly recommended for toxicologists, pharmacologists, applied mathematicians, medicinal and agricultural chemists.
Instructional objectives are the cornerstone of successful instruction. When written well, they enable you to identify appropriate content for your instruction, organize your instruction in the best way possible, and create tools to accurately determine if instruction is achieving your goals. This book is your systematic guide to identifying, selecting, and writing objectives that create the foundation for instructional success. Newly revised and completely updated, this third edition shows you how to write objectives that give you the power to: select the best content and methods for achieving your objectives; provide learners with a road map to guide them through the learning process; give learners a better chance of succeeding; and demonstrate the value of what you're teaching.
They're not doing what they should be doing - Explore fase fixes? - Are the consequences right-side up? - Are there other causes? - Which solutions are best? - Quick-reference checklist & final thoughts.
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