While drug therapies developed in the last 80 years have markedly improved treatment outcomes and the management of some types of cancers, the lack of effectiveness and side effects associated with the most common treatment types remain unacceptable. However, recent technological advances are leading to improved therapies based on targeting distinct biological pathways in cancer cells. Chemistry and Pharmacology of Anticancer Drugs is a comprehensive survey of all families of anticancer agents and therapeutic approaches currently in use or in advanced stages of clinical trials, including biological-based therapies. The book is unique in providing molecular structures for all anticancer agents, discussing them in terms of history of development, chemistry, mechanism of action, structure–function relationships, and pharmacology. It also provides relevant information on side effects, dosing, and formulation. The authors, renowned scientists in cancer research and drug discovery, also provide up-to-date information on the drug discovery process, including discussions of new research tools, tumor-targeting strategies, and fundamental concepts in the relatively new areas of precision medicine and chemoprevention. Chemistry and Pharmacology of Anticancer Drugs is an indispensable resource for cancer researchers, medicinal chemists and other biomedical scientists involved in the development of new anticancer therapies. Its breadth of coverage, clear explanations, and illustrations also make it suitable for undergraduate and postgraduate courses in medicine, pharmacy, nursing, dentistry, nutrition, the biomedical sciences, and related disciplines. Key Features: Summarizes the fundamental causes of cancer, modes of treatment, and strategies for cancer drug discovery Brings together a broad spectrum of information relating to the chemistry and pharmacology of all families of anticancer agents and therapies Includes up-to-date information on cutting-edge aspects of cancer treatments such as biomarkers, pharmacogenetics, and pharmacogenomics Features new chapters on the "Evolution of Anticancer Therapies", "Antibody-Based Therapies", and "Cancer Chemoprevention
This meticulously researched reference work documents the role of women who contributed to the development of Americanist archaeology from 1865 to 1940. Between the Civil War and World War II, many women went into anthropology and archaeology, fields that, at the beginning of this period, welcomed and made room for amateurs of both genders. But over time, the increasingly professional structure of these fields diminished or even obscured the contributions of women due to their lack of access to prestigious academic employment and publishing opportunities. As a result, a woman archaeologist during this period often published her research under her husband's name or as a junior author with her husband. In Cultural Negotiations archaeologist David L. Browman has scoured the archaeological literature and archival records of several institutions to bring the stories of more than two hundred women in Americanist archaeology to light through detailed biographies that discuss their contributions and publications. This work highlights how the social and cultural construction of archaeology as a field marginalized women and will serve as an invaluable reference to those researchers who continue to uncover the history of women in the sciences.
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