Macrolide antibiotics represent a class of natural macrocyclic products, one of the most clinically important antibiotics. Unfortunately, the production and development of new macrolide antibiotics are not represented enough in the pharmaceutical industry today. The intention of the book is therefore not only to be a teaching tool for students and experts, but also to draw the attention of the general public to this extremely useful, cheap and relatively unharmful effective anti-macrobials, and potential anti-malarials. The authors introduce the different classes of macrolides and their derivatives, principles of their biological activity, their structure and interactions with biological targets as well as synthetic methods to produce new macrolide antibiotics of similar or improved properties. Special emphasis was put on conjugates of macrolides with nucleobases or nucleosides with numerous applications; among them the most important remains the attempt to overcome bacterial resistance.
Macrolide antibiotics represent a class of natural macrocyclic products, one of the most clinically important antibiotics. Unfortunately, the production and development of new macrolide antibiotics are not represented enough in the pharmaceutical industry today. The intention of the book is therefore not only to be a teaching tool for students and experts, but also to draw the attention of the general public to this extremely useful, cheap and relatively unharmful effective anti-macrobials, and potential anti-malarials. The authors introduce the different classes of macrolides and their derivatives, principles of their biological activity, their structure and interactions with biological targets as well as synthetic methods to produce new macrolide antibiotics of similar or improved properties. Special emphasis was put on conjugates of macrolides with nucleobases or nucleosides with numerous applications; among them the most important remains the attempt to overcome bacterial resistance.
This book highlights Belgrade, reviewing its recent and historical developments and emphasizing its major ongoing planning projects. The book is divided into eight chapters. The first, entitled The urban, political and socioeconomic rise and fall of Belgrade through its history, introduces the reader to the city, and is followed by a chapter on Belgrade’s urban plans through history. The book continues with a chapter on one of the major urban projects in the former Yugoslavia, the construction of New Belgrade, its development and results, entitled New Belgrade: from no man’s land to modern city. In turn, the following three chapters explore three dominant contemporary topics: Belgrade’s riverfront redevelopment; Reimaging Belgrade: the case of Savamala; and Sustainable Belgrade. Expansion of the pedestrian zone in the city center. The book draws to a close with a chapter on Future predictions: South-Eastern European metropolis of the 21st century. This chapter in particular discusses large city projects and includes predictions about the city’s future.
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